GI-1606
I+D de fármacos
Publikationen (379) Publikationen, an denen Forscher/innen teilgenommen haben
2024
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N-(coumarin-3-yl)cinnamamide Promotes Immunomodulatory, Neuroprotective, and Lung Function-Preserving Effects during Severe Malaria
Pharmaceuticals, Vol. 17, Núm. 1
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Study of the DNA damage and cell death in human peripheral blood mononuclear and HepG2/C3A cells exposed to the synthetic 3-(3-hydroxyphenyl)-7-hydroxycoumarin
Journal of Toxicology and Environmental Health - Part A: Current Issues, Vol. 87, Núm. 1, pp. 33-46
2023
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2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 38, Núm. 1
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3D printing of a palladium-alumina cermet monolithic catalyst: catalytic evaluation in microwave-assisted cross-coupling reactions
Materials Today Chemistry, Vol. 27
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3D-Printing of Capsule Devices as Compartmentalization Tools for Supported Reagents in the Search of Antiproliferative Isatins
Pharmaceuticals, Vol. 16, Núm. 2
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8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies
European Journal of Medicinal Chemistry, Vol. 248
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Cytogenotoxicity assessment of 3-(3,4-dihydroxyphenyl)-7,8-dihydroxycoumarin on HepG2/C3A cells and leukocytes
Journal of Applied Toxicology, Vol. 43, Núm. 2, pp. 323-334
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Design of 3-Phenylcoumarins and 3-Thienylcoumarins as Potent Xanthine Oxidase Inhibitors: Synthesis, Biological Evaluation, and Docking Studies
ChemMedChem, Vol. 18, Núm. 21
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Evaluation of in vitro cytotoxic and genotoxic effects of the 3-(3,4-dihydroxyphenyl)-8-hydroxycoumarin
Journal of Applied Toxicology, Vol. 43, Núm. 10, pp. 1488-1498
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In silico approaches to develop new phenyl-pyrimidines as glycogen synthase kinase 3 (GSK-3) inhibitors with halogen-bonding capabilities: 3D-QSAR CoMFA/CoMSIA, molecular docking and molecular dynamics studies
Journal of Biomolecular Structure and Dynamics, Vol. 41, Núm. 22, pp. 13250-13259
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Modulating Cytotoxicity with Lego-like Chemistry: Upgrading Mitochondriotropic Antioxidants with Prototypical Cationic Carrier Bricks
Journal of Medicinal Chemistry, Vol. 66, Núm. 3, pp. 1835-1851
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Oxidation-labile linkers for controlled drug delivery
Bioorganic and Medicinal Chemistry Letters, Vol. 87
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Phytochemical Analysis and Antiproliferative Activity of Ulex gallii Planch. (Fabaceae), a Medicinal Plant from Galicia (Spain)
Molecules, Vol. 28, Núm. 1
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Propargylamine: an important moiety in drug discovery
Future Medicinal Chemistry, Vol. 15, Núm. 1, pp. 211-224
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Recent Advances in Biologically Active Coumarins from Marine Sources: Synthesis and Evaluation
Marine Drugs, Vol. 21, Núm. 1
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The Southern European Atlantic Diet and Its Supplements: The Chemical Bases of Its Anticancer Properties
Nutrients, Vol. 15, Núm. 19
2022
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A comprehensive ethnobotanical profile of Ocimum campechianum (Lamiaceae): from traditional medicine to phytochemical and pharmacological evidences
Plant Biosystems, Vol. 156, Núm. 6, pp. 1388-1404
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Coumarin-Resveratrol-Inspired Hybrids as Monoamine Oxidase B Inhibitors: 3-Phenylcoumarin versus trans-6-Styrylcoumarin
Molecules, Vol. 27, Núm. 3
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Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties
European Journal of Medicinal Chemistry, Vol. 239
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Hydroxy-3-Phenylcoumarins as Multitarget Compounds for Skin Aging Diseases: Synthesis, Molecular Docking and Tyrosinase, Elastase, Collagenase and Hyaluronidase Inhibition, and Sun Protection Factor
Molecules, Vol. 27, Núm. 20