Publikationen in Zusammenarbeit mit Forschern von Centre National de la Recherche Scientifique (8)

2023

  1. Corrigendum to “Lithocholic acid-based design of noncalcemic vitamin D receptor agonists” [Bioorg. Chem. 111 (2021) 104878] (Bioorganic Chemistry (2021) 111, (S0045206821002558), (10.1016/j.bioorg.2021.104878))

    Bioorganic Chemistry

2021

  1. Design, Synthesis, Evaluation and Structure of Allenic 1α,25-Dihydroxyvitamin D3 Analogs with Locked Mobility at C-17

    Chemistry - A European Journal, Vol. 27, Núm. 53, pp. 13384-13389

  2. Design, synthesis and evaluation of side-chain hydroxylated derivatives of lithocholic acid as potent agonists of the vitamin D receptor (VDR)

    Bioorganic Chemistry, Vol. 115

  3. Lithocholic acid-based design of noncalcemic vitamin D receptor agonists

    Bioorganic Chemistry, Vol. 111

2011

  1. 1α,25(OH)2-3-epi-vitamin D3, a natural physiological metabolite of vitamin D3: Its synthesis, biological activity and crystal structure with its receptor

    PLoS ONE, Vol. 6, Núm. 3

  2. Synthesis, structure, and biological activity of des-side Chain analogues of 1α,25-Dihydroxyvitamin D3 with substituents at C18

    ChemMedChem, Vol. 6, Núm. 5, pp. 788-793

2008

  1. Structure-Based Design of a Superagonist Ligand for the Vitamin D Nuclear Receptor

    Chemistry and Biology, Vol. 15, Núm. 4, pp. 383-392

2007

  1. Crystal structure of the vitamin D nuclear receptor ligand binding domain in complex with a locked side chain analog of calcitriol

    Archives of Biochemistry and Biophysics, Vol. 460, Núm. 2, pp. 172-176