Publications in collaboration with researchers from Imperial College London (15)

2023

  1. Dimeric Metal-Salphen Complexes Which Target Multimeric G-Quadruplex DNA

    Bioconjugate Chemistry, Vol. 34, Núm. 5, pp. 911-921

2021

  1. A Suite of Activity-Based Probes to Dissect the KLK Activome in Drug-Resistant Prostate Cancer

    Journal of the American Chemical Society, Vol. 143, Núm. 23, pp. 8911-8924

2020

  1. Antibody-PROTAC Conjugates Enable HER2-Dependent Targeted Protein Degradation of BRD4

    ACS Chemical Biology, Vol. 15, Núm. 6, pp. 1306-1312

  2. Hanessian-Hullar reaction in the synthesis of highly substituted trans-3,4-dihydroxypyrrolidines: Rhamnulose iminosugar mimics inhibit α-glucosidase

    Tetrahedron, Vol. 76, Núm. 1

  3. The Missing Link between (Un)druggable and Degradable KRAS

    ACS Central Science, Vol. 6, Núm. 8, pp. 1281-1284

2017

  1. Computer-aided design of multi-target ligands at A1R, A2AR and PDE10A, key proteins in neurodegenerative diseases

    Journal of Cheminformatics, Vol. 9, Núm. 1

2016

  1. 6-Deoxyhexoses from l-Rhamnose in the Search for Inducers of the Rhamnose Operon: Synergy of Chemistry and Biotechnology

    Chemistry - A European Journal, Vol. 22, Núm. 35, pp. 12557-12565

  2. Synthetic Chemical Inducers and Genetic Decoupling Enable Orthogonal Control of the rhaBAD Promoter

    ACS Synthetic Biology, Vol. 5, Núm. 10, pp. 1136-1145

2010

  1. Chiral aziridination of olefins using a chiral sulfanamide as the nitrogen source

    Synlett, pp. 145-149

1999

  1. Total synthesis of the cholesterol biosynthesis inhibitor 1233A via a (π-allyl)tricarbonyliron lactone complex

    Journal of the Chemical Society - Perkin Transactions 1, pp. 1917-1925

1988

  1. Formal synthesis of the antitumour antibiotic CC-1065

    Journal of the Chemical Society, Perkin Transactions 1, pp. 2491-2499

1987

  1. Synthesis of the combined centre- and right-hand section of the antitumour agent CC-1065

    Tetrahedron Letters, Vol. 28, Núm. 27, pp. 3163-3166

  2. Vinyl azides in heterocyclic synthesis. Part 8. Synthesis of the naturally occurring phosphodiesterase inhibitors PDE-I and PDE-II

    Journal of the Chemical Society, Perkin Transactions 1, pp. 931-935

1986

  1. Synthesis of the left-hand unit of the antitumour agent CC-1065

    Journal of the Chemical Society, Chemical Communications, pp. 1062-1063

1985

  1. Synthesis of the phosphodiesterase inhibitors PDE-I and PDE-II

    Journal of the Chemical Society, Chemical Communications, pp. 1775-1776