Publicacións nas que colabora con Abel Crespo Gavilán (12)

2022

  1. Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1Antagonists

    Journal of Medicinal Chemistry, Vol. 65, Núm. 3, pp. 2091-2106

2021

  1. 3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition

    Journal of medicinal chemistry, Vol. 64, Núm. 1, pp. 458-480

2017

  1. 3-Oxopyridazin-5-yl-Chalcone Hybrids: Potent Antiplatelet Agents That Prevent Glycoprotein IIb/IIIa Activation

    ChemistrySelect, Vol. 2, Núm. 17, pp. 4920-4933

  2. Exploring the influence of the substituent at position 4 in a series of 3,4-dihydropyrimidin-2(1H)-one A2B adenosine receptor antagonists

    Chemistry of Heterocyclic Compounds, Vol. 53, Núm. 3, pp. 316-322

2016

  1. Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes

    Journal of Medicinal Chemistry, Vol. 59, Núm. 5, pp. 1967-1983

2013

  1. Discovery of 3,4-dihydropyrimidin-2(1 H)-ones as a novel class of potent and selective A2B adenosine receptor antagonists

    ACS Medicinal Chemistry Letters, Vol. 4, Núm. 11, pp. 1031-1036

  2. Three-component assembly of structurally diverse 2-aminopyrimidine-5- carbonitriles

    ACS Combinatorial Science, Vol. 15, Núm. 7, pp. 370-378

2012

  1. Estrategias multicomponente en el descubrimiento de fármacos, identificación y optimización de antagonistas selectivos de los receptores de adenosina empleando la reacción de Biginelli

    Estrategias multicomponente en el descubrimiento de fármacos, identificación y optimización de antagonistas selectivos de los receptores de adenosina empleando la reacción de Biginelli

2011

  1. Convergent assembly of structurally diverse quinazolines

    Organic and Biomolecular Chemistry, Vol. 9, Núm. 2, pp. 351-357

  2. Supported TBD-assisted solution phase diversification of formyl-aza-heterocycles through alkylation-knoevenagel one pot sequences

    Combinatorial Chemistry and High Throughput Screening, Vol. 14, Núm. 7, pp. 570-582

2008

  1. Synthetic applications of polystyrene-supported 1,1,3,3- tetramethylguanidine

    Combinatorial Chemistry and High Throughput Screening, Vol. 11, Núm. 10, pp. 843-847

2006

  1. Pyridazines part 41: Synthesis, antiplatelet activity and SAR of 2,4,6-substituted 5-(3-oxo-3-phenylprop-1-en-1-yl)- or 5-(3-phenylprop-2-enoyl) pyridazin-3(2H)-ones

    Bioorganic and Medicinal Chemistry Letters, Vol. 16, Núm. 4, pp. 1080-1083