Publicacións nas que colabora con Miguel Maestro (42)

2023

  1. Further Studies on the Highly Active Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3 (Calcitriol): Refinement of the Side Chain

    Journal of Medicinal Chemistry, Vol. 66, Núm. 22, pp. 15326-15339

2022

  1. Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3

    Journal of Medicinal Chemistry, Vol. 65, Núm. 19, pp. 13112-13124

2021

  1. Design, Synthesis, Evaluation and Structure of Allenic 1α,25-Dihydroxyvitamin D3 Analogs with Locked Mobility at C-17

    Chemistry - A European Journal, Vol. 27, Núm. 53, pp. 13384-13389

2019

  1. Synthesis of 28,28,28-trideutero-25-hydroxydihydrotachysterol 2

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 185, pp. 248-250

  2. Mechanistic insights for the transprotection of tertiary amines with Boc2O: Via charged carbamates: Access to both enantiomers of 2-azanorbornane-3- exo -carboxylic acids

    Organic Chemistry Frontiers, Vol. 6, Núm. 20, pp. 3540-3554

2018

  1. Total synthesis of 1α,25-dihydroxyvitamin D 3 analogs modified at the side chain and D-ring

    Organic and Biomolecular Chemistry, Vol. 16, Núm. 24, pp. 4563-4569

  2. Stereoselective synthesis of 25S,26-dihydroxyvitamin D 3

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 177, pp. 247-249

  3. Aromatic-Based Design of Highly Active and Noncalcemic Vitamin D Receptor Agonists

    Journal of Medicinal Chemistry, Vol. 61, Núm. 11, pp. 4928-4937

  4. Stereoselective Palladium-Catalyzed Approach to Vitamin D3 Derivatives in Protic Medium

    Chemistry - A European Journal, Vol. 24, Núm. 13, pp. 3314-3320

  5. Synthesis of Side-Chain Locked Analogs of 1α,25-Dihydroxyvitamin D3 Bearing a C17 Methyl Group

    Organic Letters, Vol. 20, Núm. 9, pp. 2641-2644

2017

  1. A new approach to 19-nor-A-ring phosphine oxide for the convergent synthesis of 19-nor-calcitriol

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 173, pp. 86-88

  2. Total synthesis of 1α,25-dihydroxyvitamin D3 (calcitriol) through a Si-assisted allylic substitution

    Chemical Communications, Vol. 53, Núm. 58, pp. 8144-8147

2016

  1. Carborane-based design of a potent Vitamin D receptor agonist

    Chemical Science, Vol. 7, Núm. 2, pp. 1033-1037

  2. Stereoselective synthesis of 1β,25-Dihydroxyvitamin D3 and its 26,27-hexadeuterated derivative

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 164, pp. 56-58

  3. Vitamin D receptor 2016: novel ligands and structural insights

    Expert Opinion on Therapeutic Patents, Vol. 26, Núm. 11, pp. 1291-1306

2015

  1. An efficient convergent synthesis of 1α,25-dihydroxy-3-epi-vitamin D2

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 148, pp. 31-33

  2. Pit-1 inhibits BRCA1 and sensitizes human breast tumors to cisplatin and vitamin D treatment

    Oncotarget, Vol. 6, Núm. 16, pp. 14456-14471

  3. Quantitative analytical method to evaluate the metabolism of vitamin D

    Clinica Chimica Acta, Vol. 442, pp. 6-12

2014

  1. 26,26,26,27,27,27-hexadeuterated-1,25-dihydroxyvitamin D3 (1,25D-d6) as adjuvant of chemotherapy in breast cancer cell lines

    Cancers, Vol. 6, Núm. 1, pp. 67-78

  2. Clinical utility of simultaneous quantitation of 25-hydroxyvitamin D and 24,25-dihydroxyvitamin D by LC-MS/MS involving derivatization with DMEQ-TAD

    Journal of Clinical Endocrinology and Metabolism, Vol. 99, Núm. 7, pp. 2567-2574