Publicacións en colaboración con investigadores/as de University of Cagliari (51)

2023

  1. 2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms

    Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 38, Núm. 1

  2. Design of 3-Phenylcoumarins and 3-Thienylcoumarins as Potent Xanthine Oxidase Inhibitors: Synthesis, Biological Evaluation, and Docking Studies

    ChemMedChem, Vol. 18, Núm. 21

2022

  1. Coumarin-Resveratrol-Inspired Hybrids as Monoamine Oxidase B Inhibitors: 3-Phenylcoumarin versus trans-6-Styrylcoumarin

    Molecules, Vol. 27, Núm. 3

  2. Hydroxy-3-Phenylcoumarins as Multitarget Compounds for Skin Aging Diseases: Synthesis, Molecular Docking and Tyrosinase, Elastase, Collagenase and Hyaluronidase Inhibition, and Sun Protection Factor

    Molecules, Vol. 27, Núm. 20

2020

  1. Looking for new xanthine oxidase inhibitors: 3-Phenylcoumarins versus 2-phenylbenzofurans

    International Journal of Biological Macromolecules, Vol. 162, pp. 774-780

  2. Structure-Based Optimization of Coumarin hA3 Adenosine Receptor Antagonists

    Journal of Medicinal Chemistry, Vol. 63, Núm. 5, pp. 2577-2587

2019

  1. Antibacterial Activity and Molecular Docking Studies of a Selected Series of Hydroxy-3-arylcoumarins

    Molecules (Basel, Switzerland), Vol. 24, Núm. 15

  2. Discovery of new phthalazinones as vasodilator agents and novel pharmacological tools to study calcium channels

    Future Medicinal Chemistry, Vol. 11, Núm. 3, pp. 179-191

2018

  1. Coumarin derivatives as promising xanthine oxidase inhibitors

    International Journal of Biological Macromolecules, Vol. 120, pp. 1286-1293

  2. Evaluation of trypanocidal and antioxidant activities of a selected series of 3-amidocoumarins

    Medicinal Chemistry, Vol. 14, Núm. 6, pp. 573-584

  3. Targeting α -(1,4)-glucosidase in diabetes mellitus type 2: The role of new synthetic coumarins as potent inhibitors

    Current Topics in Medicinal Chemistry, Vol. 18, Núm. 27, pp. 2327-2337

2017

  1. New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies

    Bioorganic and Medicinal Chemistry, Vol. 25, Núm. 5, pp. 1687-1695

2016

  1. Progress in the development of small molecules as new human A3 adenosine receptor ligands based on the 3-thiophenylcoumarin core

    MedChemComm, Vol. 7, Núm. 5, pp. 845-852

2015

  1. Design and discovery of tyrosinase inhibitors based on a coumarin scaffold

    RSC Advances, Vol. 5, Núm. 114, pp. 94227-94235

  2. Interest of 3-arylcoumarins as xanthine oxidase inhibitors

    19TH INTERNATIONAL ELECTRONIC CONFERENCE ON SYNTHETIC ORGANIC CHEMISTRY

2014

  1. Monoamine oxidase (MAO) inhibitory activity: 3-phenylcoumarins versus 4-hydroxy-3-phenylcoumarins

    ChemMedChem, Vol. 9, Núm. 8, pp. 1672-1676

2013

  1. MAO Inhibitory Activity of 2-Arylbenzofurans versus 3-Arylcoumarins: Synthesis, invitro Study, and Docking Calculations

    ChemMedChem, Vol. 8, Núm. 6, pp. 956-966

2012

  1. 8-Substituted 3-Arylcoumarins as Potent and Selective MAO-B Inhibitors: Synthesis, Pharmacological Evaluation, and Docking Studies

    ChemMedChem, Vol. 7, Núm. 3, pp. 464-470

  2. Antitrypanosomal and antioxidant properties of 4-hydroxycoumarins derivatives

    Bioorganic and Medicinal Chemistry Letters, Vol. 22, Núm. 17, pp. 5569-5573

  3. Erratum: Synthesis and cytotoxic activity of non-naturally substituted 4-oxycoumarin derivatives (Bioorganic and Medicinal Chemistry Letters (2012) 22 (5791-5794))

    Bioorganic and Medicinal Chemistry Letters