Publicacións (283) Publicacións de María Isabel Loza García

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2025

  1. Conformational Restriction of Designer Drugs Reveals Subtype-Selective and Biased CB2Agonists with Neuroprotective Effects

    Journal of Medicinal Chemistry, Vol. 68, Núm. 16, pp. 17103-17129

  2. Copper(II) Cyclopeptides with High ROS-Mediated Cytotoxicity

    Bioconjugate Chemistry, Vol. 36, Núm. 3, pp. 500-509

  3. Design, Synthesis, and Evaluation of a New Fluorescent Ligand for the M2 Muscarinic Acetylcholine Receptor

    ACS Medicinal Chemistry Letters

  4. Design, Synthesis, and Evaluation of a New Fluorescent Ligand for the M2 Muscarinic Acetylcholine Receptor

    ACS Medicinal Chemistry Letters, Vol. 16, Núm. 4, pp. 552-559

  5. Dimethoxybenzohomoadamantane-based soluble epoxide hydrolase inhibitors: in vivo efficacy in a murine model of chemotherapy-induced neuropathic pain

    Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 40, Núm. 1

  6. Discovery of (3-Phenylcarbamoyl-3,4-dihydro-2H-pyrrol-2-yl)phosphonates as Imidazoline I2 Receptor Ligands with Anti-Alzheimer and Analgesic Properties

    Journal of Medicinal Chemistry, Vol. 68, Núm. 3, pp. 2551-2573

  7. Discovery of N-substituted-2-((arylethyl)amino)-2-(2-methoxyphenyl) acetamides: A novel family of antiplatelet agents

    Biomedicine and Pharmacotherapy, Vol. 186

  8. Distinctive patterns of G protein coupling induced by the structurally similar 5-HT2Areceptor ligands ketanserin and altanserin in human prefrontal cortex

    Molecular Pharmacology, Vol. 107, Núm. 11

  9. Exploration of JAK/STAT pathway activation in ulcerative colitis reveals sex-dependent activation of JAK2/STAT3 in the inflammatory response

    Frontiers in Immunology, Vol. 16

  10. Exploring Trisubstituted adenine derivatives as adenosine A1 receptor ligands with antagonist activity: Synthesis, biological evaluation and molecular modelling

    Bioorganic Chemistry, Vol. 159

  11. Feasibility of Multiplex Cytokine Profiling in Preterm Labor: Towards Biomarker Discovery

    Biology, Vol. 14, Núm. 6

  12. In Silico and In Vivo Pharmacological Evaluation of Iridoid Compounds: Geniposide and Asperuloside Profile Study Through Molecular Docking Assay and in the Caenorhabditis elegans Model

    Biomolecules, Vol. 15, Núm. 8

  13. Morphological profiling data resource enables prediction of chemical compound properties

    iScience, Vol. 28, Núm. 5

  14. Proline Homologation in Melanostatin Neuropeptide: Discovery of Potent Modulators of the Dopamine D<sub>2</sub> Receptors

    ACS Medicinal Chemistry Letters, Vol. 16, Núm. 8, pp. 1437-1444

  15. Rapid traversal of vast chemical space using machine learning-guided docking screens

    NATURE COMPUTATIONAL SCIENCE, Vol. 5, Núm. 4

  16. Synthesis of 2-(3-aminopropyl)benzopyrans as potential antipsychotic agents targeting D2/D3 and 5-HT2A receptors

    Bioorganic and Medicinal Chemistry, Vol. 129

  17. Warming induces unexpectedly high soil respiration in a wet tropical forest

    Nature Communications , Vol. 16, Núm. 1

2024

  1. 2-Aryladenine Derivatives as a Potent Scaffold for Adenosine Receptor Antagonists: The 6-Morpholino Derivatives

    Molecules, Vol. 29, Núm. 11

  2. Design, synthesis and validation of a new Crimped Head-Piece for DNA-Encoded libraries generation

    Bioorganic and Medicinal Chemistry, Vol. 99

  3. Effect of Bulky N-Dibenzofuranylmethyl Substitution on the 5-HT2 Receptor Affinity and Efficacy of a Psychedelic Phenethylamine

    ACS Chemical Neuroscience, Vol. 15, Núm. 3, pp. 608-616