Publicacións en colaboración con investigadores/as de University of Strasbourg (11)

2023

  1. Corrigendum to “Lithocholic acid-based design of noncalcemic vitamin D receptor agonists” [Bioorg. Chem. 111 (2021) 104878] (Bioorganic Chemistry (2021) 111, (S0045206821002558), (10.1016/j.bioorg.2021.104878))

    Bioorganic Chemistry

  2. Further Studies on the Highly Active Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3 (Calcitriol): Refinement of the Side Chain

    Journal of Medicinal Chemistry, Vol. 66, Núm. 22, pp. 15326-15339

2022

  1. Advances in Vitamin D Receptor Function and Evolution Based on the 3D Structure of the Lamprey Ligand-Binding Domain

    Journal of Medicinal Chemistry, Vol. 65, Núm. 7, pp. 5821-5829

  2. Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3

    Journal of Medicinal Chemistry, Vol. 65, Núm. 19, pp. 13112-13124

2021

  1. Design, Synthesis, Evaluation and Structure of Allenic 1α,25-Dihydroxyvitamin D3 Analogs with Locked Mobility at C-17

    Chemistry - A European Journal, Vol. 27, Núm. 53, pp. 13384-13389

  2. Design, synthesis and evaluation of side-chain hydroxylated derivatives of lithocholic acid as potent agonists of the vitamin D receptor (VDR)

    Bioorganic Chemistry, Vol. 115

  3. Lithocholic acid-based design of noncalcemic vitamin D receptor agonists

    Bioorganic Chemistry, Vol. 111

2018

  1. Aromatic-Based Design of Highly Active and Noncalcemic Vitamin D Receptor Agonists

    Journal of Medicinal Chemistry, Vol. 61, Núm. 11, pp. 4928-4937

2011

  1. 1α,25(OH)2-3-epi-vitamin D3, a natural physiological metabolite of vitamin D3: Its synthesis, biological activity and crystal structure with its receptor

    PLoS ONE, Vol. 6, Núm. 3

2010

  1. Structure-function relationships and crystal structures of the vitamin D receptor bound 2α-methyl-(20S,23S)- and 2α-methyl-(20S,23R)- epoxymethano-1α,25-dihydroxyvitamin D3

    Journal of Medicinal Chemistry, Vol. 53, Núm. 3, pp. 1159-1171

2007

  1. Crystal structure of the vitamin D nuclear receptor ligand binding domain in complex with a locked side chain analog of calcitriol

    Archives of Biochemistry and Biophysics, Vol. 460, Núm. 2, pp. 172-176