Publications by the researcher in collaboration with JOSE ANGEL FONTENLA GIL (17)

2023

  1. 8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies

    European Journal of Medicinal Chemistry, Vol. 248

2021

  1. Gamma-decanolactone: Preliminary evaluation as potential antiparkinsonian drug

    European Journal of Pharmacology, Vol. 906

2003

  1. New arylpiperazine derivatives with high affinity for α1A, D2 and 5-HT2A receptors

    Bioorganic and Medicinal Chemistry Letters, Vol. 13, Núm. 2, pp. 175-178

2000

  1. Butyrophenone analogues in the carbazole series as potential atypical antipsychotics: Synthesis and determination of affinities at D2, 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors

    European Journal of Medicinal Chemistry, Vol. 35, Núm. 1, pp. 83-95

  2. Conformationally constrained butyrophenones with affinity for dopamine (D1, D2, D4) and serotonin (5-HT(2A), 5-HT(2B), 5-HT(2C)) receptors: Synthesis of aminomethylbenzo[b]furanones and their evaluation as antipsychotics

    Journal of Medicinal Chemistry, Vol. 43, Núm. 24, pp. 4678-4693

1999

  1. Conformationally constrained butyrophenones with mixed dopaminergic (D2) and serotoninergic (5-HT2(A), 5-HT2(C)) affinities: Synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo- and - thienocycloalkanones as putative atypical antipsychotics

    Journal of Medicinal Chemistry, Vol. 42, Núm. 15, pp. 2774-2797

1998

  1. Butyrophenone analogues in the carbazole series: Synthesis and determination of affinities at D2 and 5-HT(2A) receptors

    Bioorganic and Medicinal Chemistry Letters, Vol. 8, Núm. 24, pp. 3571-3576

1997

  1. New cyclic butyrophenone derivatives in the indole series as potential atypical antipsychotics. A simple and practical synthesis of 6-aminomethyl-tetrahydroindol-4-ones and their affinities for D2 and 5-HT(2A) receptors

    Bioorganic and Medicinal Chemistry Letters, Vol. 7, Núm. 7, pp. 913-918

1996

  1. Synthesis and affinities for dopamine (D2) and 5-hydroxytryptamine (5-HT2A) receptors of 1-(benzoylpropyl)-4-(1-oxocycloalkyl-2-ethyl)-piperazines as cyclic butyrophenone derivatives

    Chemical and Pharmaceutical Bulletin, Vol. 44, Núm. 3, pp. 534-541

1995

  1. Butyrophenone analogues: Synthesis of 2-methyl-3-ethyl-5-aminoethyl-4,5,6,7-tetrahydroindol-4-ones, and their affinities for d 1 , d 2 and 5-ht 2a receptors

    Bioorganic and Medicinal Chemistry Letters, Vol. 5, Núm. 6, pp. 579-584

1994

  1. Pyridazine derivatives XII. Synthesis and antipsychotic-antidepressant activity of some butyrophenone derivatives of 6-phenylpyridazine

    European Journal of Medicinal Chemistry, Vol. 29, Núm. 11, pp. 831-839

  2. Synthesis and Atypical Antipsychotic Profile of Some 2-(2-Piperidinoethyl)benzocycloalkanones as Analogs of Butyrophenone

    Journal of Medicinal Chemistry, Vol. 37, Núm. 16, pp. 2564-2573

1993

  1. Antiserotoninergic activity of 2‐aminoethylbenzocyclanones in rat aorta: Structure‐activity relationships

    Journal of Pharmaceutical Sciences, Vol. 82, Núm. 5, pp. 513-517

  2. Cyproheptadine analogues: Synthesis, antiserotoninergic activity, and structure‐activity relationships

    Journal of Pharmaceutical Sciences, Vol. 82, Núm. 11, pp. 1090-1093

1992

  1. Effect of urethane on hydralazine-induced tachycardia in rats

    General Pharmacology, Vol. 23, Núm. 6, pp. 1143-1147

1991

  1. 5-HT2 antagonist activity of 3-aminomethyltetralones

    Bioorganic and Medicinal Chemistry Letters, Vol. 1, Núm. 12, pp. 717-720

1984

  1. SINTESIS Y ESTUDIO DE LA POSIBLE ACTIVIDAD NEUROLEPTICA DEL 3-(p-FLUOROBENZOIL)-TROPANO

    Archivos de Farmacologia y Toxicologia, Vol. 10, Núm. 3, pp. 151-160