Publications by the researcher in collaboration with RITA SIGUEIRO PONTE (22)

2019

  1. Synthesis of 28,28,28-trideutero-25-hydroxydihydrotachysterol 2

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 185, pp. 248-250

2018

  1. Stereoselective synthesis of 25S,26-dihydroxyvitamin D 3

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 177, pp. 247-249

  2. Aromatic-Based Design of Highly Active and Noncalcemic Vitamin D Receptor Agonists

    Journal of Medicinal Chemistry, Vol. 61, Núm. 11, pp. 4928-4937

  3. Stereoselective Palladium-Catalyzed Approach to Vitamin D3 Derivatives in Protic Medium

    Chemistry - A European Journal, Vol. 24, Núm. 13, pp. 3314-3320

  4. Studies on the synthesis of vitamin D analogs with aromatic D-ring

    Anais da Academia Brasileira de Ciencias, Vol. 90, Núm. 1, pp. 1035-1042

  5. Synthesis of Side-Chain Locked Analogs of 1α,25-Dihydroxyvitamin D3 Bearing a C17 Methyl Group

    Organic Letters, Vol. 20, Núm. 9, pp. 2641-2644

2017

  1. A new approach to 19-nor-A-ring phosphine oxide for the convergent synthesis of 19-nor-calcitriol

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 173, pp. 86-88

2016

  1. Carborane-based design of a potent Vitamin D receptor agonist

    Chemical Science, Vol. 7, Núm. 2, pp. 1033-1037

  2. Stereoselective synthesis of 1β,25-Dihydroxyvitamin D3 and its 26,27-hexadeuterated derivative

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 164, pp. 56-58

2015

  1. An efficient convergent synthesis of 1α,25-dihydroxy-3-epi-vitamin D2

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 148, pp. 31-33

  2. Pit-1 inhibits BRCA1 and sensitizes human breast tumors to cisplatin and vitamin D treatment

    Oncotarget, Vol. 6, Núm. 16, pp. 14456-14471

2014

  1. Clinical utility of simultaneous quantitation of 25-hydroxyvitamin D and 24,25-dihydroxyvitamin D by LC-MS/MS involving derivatization with DMEQ-TAD

    Journal of Clinical Endocrinology and Metabolism, Vol. 99, Núm. 7, pp. 2567-2574

  2. Synthesis of nonadeuterated 1α,25-dihydroxyvitamin D2

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 144, Núm. PART A, pp. 204-206

2013

  1. Metabolic stability of 3-Epi-1α,25-dihydroxyvitamin D3 over 1 α 25-dihydroxyvitamin D3: Metabolism and molecular docking studies using rat CYP24A1

    Journal of Cellular Biochemistry, Vol. 114, Núm. 10, pp. 2293-2305

  2. Synthesis of 9-alkylated calcitriol and two 1α,25-dihydroxy-9- methylene-10,19-dihydrovitamin D3 analogues with a non-natural triene system by thermal sigmatropic rearrangements

    Journal of Organic Chemistry, Vol. 78, Núm. 4, pp. 1444-1450

2011

  1. 1α,25(OH)2-3-epi-vitamin D3, a natural physiological metabolite of vitamin D3: Its synthesis, biological activity and crystal structure with its receptor

    PLoS ONE, Vol. 6, Núm. 3

2010

  1. An expeditious route to 1α,25-dihydroxyvitamin D3 and its analogues by an aqueous tandem palladium-catalyzed a-ring closure and suzuki coupling to the C/D unit

    Chemistry - A European Journal, Vol. 16, Núm. 5, pp. 1432-1435

  2. Design and synthesis of active vitamin D analogs

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 121, Núm. 1-2, pp. 7-12

  3. Structure-function relationships and crystal structures of the vitamin D receptor bound 2α-methyl-(20S,23S)- and 2α-methyl-(20S,23R)- epoxymethano-1α,25-dihydroxyvitamin D3

    Journal of Medicinal Chemistry, Vol. 53, Núm. 3, pp. 1159-1171

  4. Synthesis and biological evaluation of 6-methyl analog of 1α,25-dihydroxyvitamin D3

    Journal of Steroid Biochemistry and Molecular Biology, Vol. 121, Núm. 1-2, pp. 29-33