Discovery of New Potent Positive Allosteric Modulators of Dopamine D2Receptors: Insights into the Bioisosteric Replacement of Proline to 3-Furoic Acid in the Melanostatin Neuropeptide

  1. Sampaio-Dias, I.E.
  2. Reis-Mendes, A.
  3. Costa, V.M.
  4. García-Mera, X.
  5. Brea, J.
  6. Loza, M.I.
  7. Pires-Lima, B.L.
  8. Alcoholado, C.
  9. Algarra, M.
  10. Rodríguez-Borges, J.E.
Revista:
Journal of Medicinal Chemistry

ISSN: 1520-4804 0022-2623

Ano de publicación: 2021

Volume: 64

Número: 9

Páxinas: 6209-6220

Tipo: Artigo

DOI: 10.1021/ACS.JMEDCHEM.1C00252 GOOGLE SCHOLAR