Discovery of a novel class of potent coumarin monoamine oxidase B inhibitors: Development and biopharmacological profiling of 7-[(3-chlorobenzyl) oxy]-4-[(methylamino)methyl]-2H-chromen-2-one methanesulfonate (NW-1772) as a highly potent, selective, reversible, and orally active monoamine oxidase B inhibitor

  1. Pisani, L.
  2. Muncipinto, G.
  3. Miscioscia, T.F.
  4. Nicolotti, O.
  5. Leonetti, F.
  6. Catto, M.
  7. Caccia, C.
  8. Salvati, P.
  9. Soto-Otero, R.
  10. Mendez-Alvarez, E.
  11. Passeleu, C.
  12. Carotti, A.
Revista:
Journal of Medicinal Chemistry

ISSN: 0022-2623

Ano de publicación: 2009

Volume: 52

Número: 21

Páxinas: 6685-6706

Tipo: Artigo

DOI: 10.1021/JM9010127 GOOGLE SCHOLAR