Discovery and characterization of 4′-(2-furyl)-N-pyridin-3-yl-4, 5′-bipyrimidin-2′-amine (LAS38096), a potent, selective, and efficacious A2B adenosine receptor antagonist

  1. Vidal, B.
  2. Nueda, A.
  3. Esteve, C.
  4. Domenech, T.
  5. Benito, S.
  6. Reinoso, R.F.
  7. Pont, M.
  8. Calbet, M.
  9. López, R.
  10. Cadavid, M.I.
  11. Loza, M.I.
  12. Cárdenas, Á.
  13. Godessart, N.
  14. Beleta, J.
  15. Warrellow, G.
  16. Ryder, H.
Journal:
Journal of Medicinal Chemistry

ISSN: 0022-2623

Year of publication: 2007

Volume: 50

Issue: 11

Pages: 2732-2736

Type: Article

DOI: 10.1021/JM061333V GOOGLE SCHOLAR