INCTB
Inhibidores Enzimáticos e Ferramentas Químicas en Bioloxía
Publicacións (9) Publicacións nas que participase algún/ha investigador/a Ver datos de investigación referenciados.
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Drug Discovery
2024
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High-affinity A/T-rich DNA binding with a dimeric bisbenzamidine
NAR Molecular Medicine, Vol. 1, Núm. 4
2023
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Dimeric Metal-Salphen Complexes Which Target Multimeric G-Quadruplex DNA
Bioconjugate Chemistry, Vol. 34, Núm. 5, pp. 911-921
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Quinate-based ligands for irreversible inactivation of the bacterial virulence factor DHQ1 enzyme—A molecular insight †
Frontiers in Molecular Biosciences, Vol. 10
2022
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Regioselective Synthesis of 2-Aryl-5-cyano-1-(2-hydroxyaryl)-1 H-imidazole-4-carboxamides Self-Assisted by a 2-Hydroxyaryl Group
ACS Omega, Vol. 7, Núm. 27, pp. 23289-23301
2021
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Crambescin C1 Acts as A Possible Substrate of iNOS and eNOS Increasing Nitric Oxide Production and Inducing In Vivo Hypotensive Effect
Frontiers in Pharmacology, Vol. 12
2019
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Hydroxylammonium derivatives for selective active-site lysine modification in the anti-virulence bacterial target DHQ1 enzyme
Organic Chemistry Frontiers, Vol. 6, Núm. 17, pp. 3127-3135
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Synthesis of rigidified shikimic acid derivatives by ring-closing metathesis to imprint inhibitor efficacy against shikimate kinase enzyme
Organic Chemistry Frontiers, Vol. 6, Núm. 14, pp. 2514-2528
2018
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Photogeneration of Quinone Methides as Latent Electrophiles for Lysine Targeting
Journal of Organic Chemistry, Vol. 83, Núm. 21, pp. 13019-13029
2017
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A New Pathway for Protein Haptenation by β-Lactams
Chemistry - A European Journal, Vol. 23, Núm. 56, pp. 13986-13994